10–15 May 2026
Casino Conference Centre
Europe/Prague timezone

Synthesis of Phosphorylated Peptides Using (py)2PO2[OTf] and Their Interaction with f-Elements

14 May 2026, 17:18
3m
Gallery

Gallery

Poster Radionuclides in the Environment, Radioecology Environmental Radioactivity

Speaker

Tom Pfandt (TU Dresden)

Description

Uranium and rare earth mining, the extensive use of mineral fertilizers, nuclear weapons programs, and reprocessing plants have released significant amounts of lanthanides and actinides worldwide. The environmental contamination with f-elements can pose severe health risks, especially if they enter the human food chain. Hence, a deeper understanding of the interaction of f-elements with biochemical motifs is crucial for risk assessment and hazard management.

Studies on metalloproteins like transferrin, calmodulin, and siderocalin have revealed strong interactions with f-elements. Particularly high affinities are found for phosphoproteins like casein or phosvitin, which contain high levels of phosphoserine residues. For a detailed understanding of the binding modes and preferred coordination sites in amino acid/peptide-f-element systems, systematic investigations remain essential.

With this aim, the novel phosphorylation agent (py)2PO2[OTf] (py = pyridine, OTf = triflate) was used to functionalize dipeptides to obtain a library of bio-inspired model compounds. Their interactions with f-elements were subsequently studied. Systems of the unmodified dipeptides as well as the model compounds were investigated in combination with various Ln(III) and uranyl(VI) ions in solution using heteronuclear NMR and fluorescence spectroscopy. The results, including complex stoichiometries and identified coordination sites, are presented.

Author

Tom Pfandt (TU Dresden)

Co-authors

Prof. Jan J. Weigand (TU Dresden) Dr Marco Wenzel (TU Dresden)

Presentation materials

There are no materials yet.